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Asenapine maleate

CAS No. 85650-56-2

Asenapine maleate ( Org 5222 maleate;Org-5222 maleate;Org5222 maleate )

Catalog No. M16209 CAS No. 85650-56-2

Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 27 In Stock
10MG 42 In Stock
25MG 66 In Stock
50MG 87 In Stock
100MG 123 In Stock
200MG 213 In Stock
500MG 353 In Stock
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Biological Information

  • Product Name
    Asenapine maleate
  • Note
    Research use only, not for human use.
  • Brief Description
    Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
  • Description
    Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors; shows much lower affinity (pKi<5) for muscarinic receptor; behaves as a potent antagonist 5-HT receptors (5-HT2A pKB=9.0), dopaime and adrenoceptors; shows strong antipsychotic potential in vivo.Schizophrenia Approved
  • Synonyms
    Org 5222 maleate;Org-5222 maleate;Org5222 maleate
  • Pathway
    Angiogenesis
  • Target
    Adrenergic Receptor
  • Recptor
    5-HT2A;5-HT2B;5-HT2C;5-HT6;5-HT7
  • Research Area
    Neurological Disease
  • Indication
    Schizophrenia

Chemical Information

  • CAS Number
    85650-56-2
  • Formula Weight
    401.84
  • Molecular Formula
    C21H20ClNO5
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CN1C[C@H]2[C@H](C1)C3=C(C=CC(=C3)Cl)OC4=CC=CC=C24.C(=C\C(=O)O)\C(=O)O
  • Chemical Name
    1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Room P, et al. Eur J Pharmacol. 1991 Dec 3;205(3):233-40.
2. Broekkamp CL, et al. Arzneimittelforschung. 1990 May;40(5):544-9.
3. Psychopharmacology (Berl). 2008 Feb;196(3):417-29.
4. Shahid M, et al. J Psychopharmacol. 2009 Jan;23(1):65-73.
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